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metadata
language: []
pretty_name: AQSOL
config_name: aqsol
dataset_size: 597796
size_categories: 10K<n<100K
license: cc-by-nc-sa-4.0
license_link: https://creativecommons.org/licenses/by-nc-sa/4.0/
tags:
  - graphs
  - molecules
  - chemistry
task_categories:
  - graph-regression
homepage: https://pubs.acs.org/doi/10.1021/ci3003352

aqsol

AQSOL molecular graphs with categorical atom/bond encodings for aqueous solubility regression.

License: CC BY-NC-SA 4.0

Splits

Split Rows File Size (MB)
train 7,836 train.parquet 0.40
validation 998 val.parquet 0.08
test 999 test.parquet 0.12

Features

  • mol_id: int64 unique identifier per molecule
  • x: list[int64], shape (num_nodes,), atomic type categorical index
  • edge_index: int64[2, num_edges], COO adjacency
  • edge_attr: list[int64], shape (num_edges,), bond type categorical index
  • num_nodes: int64 number of atoms
  • y: float32 graph-level target (LogS)

Citation

@article{sorkun2019aqsol,
  title={AQSOL: A Complete Aqueous Solubility Dataset for Small Molecules},
  author={Sorkun, Murat C and Khetan, Aditya and Er, Sanli},
  journal={Journal of Cheminformatics},
  volume={11},
  number={1},
  pages={1--16},
  year={2019},
  publisher={Springer}
}