broad_id
string | depmap_id
string | ccle_name
string | screen_id
string | upper_limit
int64 | lower_limit
float64 | slope
float64 | r2
float64 | auc
float64 | ec50
float64 | ic50
float64 | name
string | moa
string | target
string | disease.area
string | indication
string | smiles
string | phase
string | passed_str_profiling
bool | row_name
string |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
BRD-K19388745-003-01-7
|
ACH-000123
|
COV434_OVARY
|
HTS002
| 1 | 2.076535 | -0.116246 | 0.050216 | 1.437137 | 0.002723 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000123
|
BRD-K19388745-003-01-7
|
ACH-000717
|
COLO680N_OESOPHAGUS
|
HTS002
| 1 | 1.495756 | -1.157578 | 0.380303 | 1.369965 | 0.897244 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000717
|
BRD-K19388745-003-01-7
|
ACH-000669
|
SW900_LUNG
|
HTS002
| 1 | 1.645408 | -0.380427 | 0.214005 | 1.278916 | 0.031462 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000669
|
BRD-K19388745-003-01-7
|
ACH-000764
|
SH10TC_STOMACH
|
HTS002
| 1 | 0.58936 | 4.266432 | 0.058664 | 0.943169 | 2.612583 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000764
|
BRD-K19388745-003-01-7
|
ACH-000288
|
BT549_BREAST
|
HTS002
| 1 | 1.448039 | -3.289555 | 0.419038 | 1.25471 | 0.151873 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000288
|
BRD-K19388745-003-01-7
|
ACH-000415
|
BICR6_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 1.033337 | 0.035997 | -0.067409 | 1.01776 | 0.002024 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000415
|
BRD-K19388745-003-01-7
|
ACH-000977
|
LNCAPCLONEFGC_PROSTATE
|
HTS002
| 1 | 1.313379 | -0.615472 | -0.154452 | 1.225174 | 0.890077 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000977
|
BRD-K19388745-003-01-7
|
ACH-000397
|
TEN_ENDOMETRIUM
|
HTS002
| 1 | 2.452274 | 0.028319 | -0.033991 | 1.713406 | 0.270043 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000397
|
BRD-K19388745-003-01-7
|
ACH-000565
|
RCM1_LARGE_INTESTINE
|
HTS002
| 1 | 2.024106 | -0.922703 | 0.396561 | 1.356744 | 0.01713 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000565
|
BRD-K19388745-003-01-7
|
ACH-000209
|
SNU1079_BILIARY_TRACT
|
HTS002
| 1 | 2.441836 | -1.683939 | 0.450762 | 1.240487 | 0.002958 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000209
|
BRD-K19388745-003-01-7
|
ACH-000927
|
BT474_BREAST
|
HTS002
| 1 | 2.321794 | 0.170956 | -0.026697 | 1.450785 | 4.544777 | null |
colforsin-daproate
|
adenylyl cyclase activator
| null | null | null |
CN(C)CCC(=O)O[C@@H]1[C@H](OC(C)=O)[C@@]2(C)O[C@](C)(CC(=O)[C@]2(O)[C@@]2(C)[C@@H](O)CCC(C)(C)[C@H]12)C=C
|
Launched
| true |
ACH-000927
|
BRD-K11640013-236-10-1
|
ACH-000879
|
MFE296_ENDOMETRIUM
|
HTS002
| 1 | 2.478067 | -0.066867 | -0.022571 | 1.70874 | 0.022665 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000879
|
BRD-K11640013-236-10-1
|
ACH-000320
|
PSN1_PANCREAS
|
HTS002
| 1 | 2.323588 | -0.057336 | -0.004279 | 1.666244 | 0.098927 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000320
|
BRD-K11640013-236-10-1
|
ACH-001145
|
OC316_OVARY
|
HTS002
| 1 | 2.479681 | -0.234177 | 0.007067 | 1.604775 | 0.013699 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-001145
|
BRD-K11640013-236-10-1
|
ACH-000873
|
KYSE270_OESOPHAGUS
|
HTS002
| 1 | 1.745582 | -0.306875 | 0.424763 | 1.370262 | 0.074158 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000873
|
BRD-K11640013-236-10-1
|
ACH-000855
|
KYSE150_OESOPHAGUS
|
HTS002
| 1 | 1.75174 | 0.061502 | 0.029839 | 1.435651 | 0.000408 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000855
|
BRD-K11640013-236-10-1
|
ACH-000913
|
ESS1_ENDOMETRIUM
|
HTS002
| 1 | 3.532497 | -0.189588 | 0.370306 | 2.016403 | 0.008203 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000913
|
BRD-K11640013-236-10-1
|
ACH-000488
|
TE11_OESOPHAGUS
|
HTS002
| 1 | 1.696469 | -0.07456 | 0.060172 | 1.342693 | 0.050744 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000488
|
BRD-K11640013-236-10-1
|
ACH-000832
|
CAL27_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 2.576791 | -0.128633 | 0.045476 | 1.530156 | 0.000335 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000832
|
BRD-K11640013-236-10-1
|
ACH-000781
|
NCIH2023_LUNG
|
HTS002
| 1 | 1.988635 | 0.119557 | -0.025989 | 1.515108 | 0.037891 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000781
|
BRD-K11640013-236-10-1
|
ACH-000137
|
8MGBA_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 2.030591 | -1.138112 | 0.583648 | 1.425037 | 0.033131 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000137
|
BRD-K11640013-236-10-1
|
ACH-000632
|
HS944T_SKIN
|
HTS002
| 1 | 4.050331 | -0.207621 | -0.125424 | 1.589882 | 0.000049 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000632
|
BRD-K11640013-236-10-1
|
ACH-000319
|
MPP89_PLEURA
|
HTS002
| 1 | 2.234776 | 0.106042 | -0.088321 | 1.664949 | 0.017647 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000319
|
BRD-K11640013-236-10-1
|
ACH-000630
|
YD8_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 1.662899 | -0.010046 | -0.010125 | 1.361464 | 5,558,716.882988 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000630
|
BRD-K11640013-236-10-1
|
ACH-000266
|
SNU213_PANCREAS
|
HTS002
| 1 | 2.08075 | -0.053783 | -0.027021 | 1.531067 | 0.041021 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000266
|
BRD-K11640013-236-10-1
|
ACH-000047
|
GCIY_STOMACH
|
HTS002
| 1 | 2.352357 | -0.769939 | 0.330142 | 1.210522 | 0.001703 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000047
|
BRD-K11640013-236-10-1
|
ACH-000273
|
SF539_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 5.47365 | -0.793399 | -0.264683 | 1.073938 | 0.000049 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000273
|
BRD-K11640013-236-10-1
|
ACH-000682
|
SNU1066_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 0.590701 | 0.388577 | -0.099863 | 0.869655 | 0.931151 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000682
|
BRD-K11640013-236-10-1
|
ACH-000359
|
MG63_BONE
|
HTS002
| 1 | 0.780436 | -0.061427 | -0.028025 | 0.847978 | 46,635.484173 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000359
|
BRD-K11640013-236-10-1
|
ACH-000846
|
FADU_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | -2.01814 | 0.287431 | 0.055332 | 0.974775 | 71,408.306569 | 257.65849 |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000846
|
BRD-K11640013-236-10-1
|
ACH-000804
|
NB1_AUTONOMIC_GANGLIA
|
HTS002
| 1 | 0.981615 | -0.217261 | -0.0151 | 0.982813 | 33,809.585503 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000804
|
BRD-K11640013-236-10-1
|
ACH-000609
|
SF126_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 0.829883 | -0.154284 | -0.023354 | 0.900351 | 0.818109 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000609
|
BRD-K11640013-236-10-1
|
ACH-000974
|
SNGM_ENDOMETRIUM
|
HTS002
| 1 | 2.22528 | 0.228811 | -0.093988 | 1.229448 | 82.450126 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000974
|
BRD-K11640013-236-10-1
|
ACH-000987
|
MEWO_SKIN
|
HTS002
| 1 | 1.380445 | 0.187366 | -0.090295 | 1.105419 | 18.010293 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000987
|
BRD-K11640013-236-10-1
|
ACH-000787
|
LXF289_LUNG
|
HTS002
| 1 | 1.696465 | 0.429453 | 0.078688 | 1.314029 | 0.144281 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000787
|
BRD-K11640013-236-10-1
|
ACH-000561
|
TT_OESOPHAGUS
|
HTS002
| 1 | 1.743412 | -0.086981 | 0.112242 | 1.369494 | 0.067996 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000561
|
BRD-K11640013-236-10-1
|
ACH-000212
|
CAL120_BREAST
|
HTS002
| 1 | 1.928065 | -0.027656 | -0.086491 | 1.599908 | 240,109,010.846349 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000212
|
BRD-K11640013-236-10-1
|
ACH-000305
|
ECGI10_OESOPHAGUS
|
HTS002
| 1 | 1.936822 | 0.065182 | 0.001648 | 1.497186 | 0.01165 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000305
|
BRD-K11640013-236-10-1
|
ACH-000138
|
CFPAC1_PANCREAS
|
HTS002
| 1 | 1.694604 | -0.175515 | -0.068787 | 1.248263 | 0.002276 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000138
|
BRD-K11640013-236-10-1
|
ACH-000250
|
KMRC20_KIDNEY
|
HTS002
| 1 | 4.12425 | 5.564644 | 0.094501 | 1.010044 | 13.483033 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000250
|
BRD-K11640013-236-10-1
|
ACH-000856
|
CAL51_BREAST
|
HTS002
| 1 | 2.612731 | 0.098965 | -0.077571 | 1.523019 | 148.956476 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000856
|
BRD-K11640013-236-10-1
|
ACH-000046
|
ACHN_KIDNEY
|
HTS002
| 1 | 1.724415 | 0.166273 | -0.083285 | 1.428709 | 0.007434 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000046
|
BRD-K11640013-236-10-1
|
ACH-000878
|
HCC15_LUNG
|
HTS002
| 1 | 1.296517 | -0.04526 | -0.028363 | 1.221802 | 2,355,295,105.39784 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000878
|
BRD-K11640013-236-10-1
|
ACH-000766
|
NCIH1648_LUNG
|
HTS002
| 1 | 1.251269 | 0.10048 | -0.043227 | 1.174074 | 0.000021 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000766
|
BRD-K11640013-236-10-1
|
ACH-000666
|
NCIH1355_LUNG
|
HTS002
| 1 | 2.178067 | -0.020025 | -0.049289 | 1.636164 | 236.35233 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000666
|
BRD-K11640013-236-10-1
|
ACH-000701
|
RMUGS_OVARY
|
HTS002
| 1 | 2.462779 | -0.282635 | 0.005275 | 1.682105 | 0.045072 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000701
|
BRD-K11640013-236-10-1
|
ACH-000884
|
MDAMB435S_SKIN
|
HTS002
| 1 | 1.787585 | -0.175088 | 0.056135 | 1.293905 | 0.003401 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000884
|
BRD-K11640013-236-10-1
|
ACH-000037
|
S117_SOFT_TISSUE
|
HTS002
| 1 | 2.114309 | -2.931453 | 0.292497 | 1.566053 | 0.084419 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000037
|
BRD-K11640013-236-10-1
|
ACH-000504
|
SNB75_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.671702 | -0.105976 | -0.046094 | 1.407848 | 5.200158 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000504
|
BRD-K11640013-236-10-1
|
ACH-000502
|
TCCPAN2_PANCREAS
|
HTS002
| 1 | 1.890219 | -0.298304 | 0.079165 | 1.338668 | 0.011626 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000502
|
BRD-K11640013-236-10-1
|
ACH-000886
|
NCIH2009_LUNG
|
HTS002
| 1 | 3.016475 | -0.265028 | 0.191376 | 1.795585 | 0.012543 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000886
|
BRD-K11640013-236-10-1
|
ACH-000035
|
NCIH1650_LUNG
|
HTS002
| 1 | 1.899733 | -0.268329 | 0.047305 | 1.413165 | 0.039068 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000035
|
BRD-K11640013-236-10-1
|
ACH-000661
|
WM1799_SKIN
|
HTS002
| 1 | 1.632509 | -0.784323 | -0.04303 | 1.07332 | 0.000953 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000661
|
BRD-K11640013-236-10-1
|
ACH-000391
|
MHHES1_BONE
|
HTS002
| 1 | 2.293779 | -0.266788 | -0.056251 | 1.721484 | 0.209357 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000391
|
BRD-K11640013-236-10-1
|
ACH-000843
|
HARA_LUNG
|
HTS002
| 1 | 1.979374 | 0.085265 | -0.026877 | 1.499729 | 0.047961 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000843
|
BRD-K11640013-236-10-1
|
ACH-000711
|
JIMT1_BREAST
|
HTS002
| 1 | 2.021596 | -0.12004 | -0.114218 | 1.730769 | 205.938012 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000711
|
BRD-K11640013-236-10-1
|
ACH-000232
|
U251MG_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 2.095483 | -0.111251 | 0.155162 | 1.55837 | 0.111676 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000232
|
BRD-K11640013-236-10-1
|
ACH-000322
|
HT144_SKIN
|
HTS002
| 1 | 2.61708 | -0.060095 | 0.067568 | 1.793275 | 0.04149 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000322
|
BRD-K11640013-236-10-1
|
ACH-000736
|
SNU601_STOMACH
|
HTS002
| 1 | 1.643364 | -0.192379 | 0.038399 | 1.380874 | 0.620271 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000736
|
BRD-K11640013-236-10-1
|
ACH-000809
|
KYSE410_OESOPHAGUS
|
HTS002
| 1 | 1.659377 | -0.117164 | -0.30057 | 1.342718 | 0.15623 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000809
|
BRD-K11640013-236-10-1
|
ACH-000747
|
NCIH1703_LUNG
|
HTS002
| 1 | 2.117766 | -0.177088 | -0.124154 | 1.467674 | 0.010876 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000747
|
BRD-K11640013-236-10-1
|
ACH-000364
|
U2OS_BONE
|
HTS002
| 1 | 3.055135 | -0.129591 | 0.006421 | 1.918658 | 0.014337 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000364
|
BRD-K11640013-236-10-1
|
ACH-000679
|
OE19_OESOPHAGUS
|
HTS002
| 1 | 1.886314 | 0.058487 | -0.012382 | 1.396617 | 2.941877 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000679
|
BRD-K11640013-236-10-1
|
ACH-000985
|
LS411N_LARGE_INTESTINE
|
HTS002
| 1 | 1.018857 | -0.312188 | -0.010553 | 1.00774 | 0.019834 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000985
|
BRD-K11640013-236-10-1
|
ACH-000441
|
SH4_SKIN
|
HTS002
| 1 | 1.844138 | -0.216836 | 0.03742 | 1.483233 | 0.338809 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000441
|
BRD-K11640013-236-10-1
|
ACH-001113
|
LC1SQSF_LUNG
|
HTS002
| 1 | 2.482744 | -0.093893 | 0.068738 | 1.697695 | 0.021765 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-001113
|
BRD-K11640013-236-10-1
|
ACH-000620
|
JHH1_LIVER
|
HTS002
| 1 | 1.820282 | 0.161747 | -0.10617 | 1.371009 | 0.270857 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000620
|
BRD-K11640013-236-10-1
|
ACH-000853
|
NCIH661_LUNG
|
HTS002
| 1 | 1.432977 | 0.388043 | 0.089869 | 1.343476 | 0.001064 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000853
|
BRD-K11640013-236-10-1
|
ACH-000102
|
GMS10_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 2.363896 | -0.209469 | 0.093013 | 1.397315 | 0.000801 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000102
|
BRD-K11640013-236-10-1
|
ACH-000648
|
NCIH28_PLEURA
|
HTS002
| 1 | 1.189011 | 0.086446 | -0.217694 | 1.122037 | 0.000068 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000648
|
BRD-K11640013-236-10-1
| null | null |
HTS002
| 1 | 1.061538 | 0.365793 | -0.071511 | 1.049511 | 0.00072 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| false |
ACH-000925_FAILED_STR
|
BRD-K11640013-236-10-1
|
ACH-001239
|
WM2664_SKIN
|
HTS002
| 1 | 1.38762 | -3.156109 | 0.262487 | 1.114454 | 0.010714 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-001239
|
BRD-K11640013-236-10-1
|
ACH-001321
|
TT_THYROID
|
HTS002
| 1 | 1.745118 | -0.399666 | 0.17826 | 1.295894 | 0.02029 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-001321
|
BRD-K11640013-236-10-1
|
ACH-000172
|
TM87_SOFT_TISSUE
|
HTS002
| 1 | 1.572646 | -1.103583 | -0.092388 | 1.16003 | 0.008775 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000172
|
BRD-K11640013-236-10-1
|
ACH-001128
|
MON_SOFT_TISSUE
|
HTS002
| 1 | 2.50075 | 0.154182 | 0.00753 | 1.746452 | 0.083869 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-001128
|
BRD-K11640013-236-10-1
|
ACH-000437
|
SW1088_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 2.286114 | 0.058907 | -0.026323 | 1.692991 | 0.005466 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000437
|
BRD-K11640013-236-10-1
|
ACH-000735
|
PECAPJ49_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 2.221663 | 0.028179 | -0.050654 | 1.654084 | 0.000505 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000735
|
BRD-K11640013-236-10-1
|
ACH-000643
|
HDQP1_BREAST
|
HTS002
| 1 | 1.718777 | 0.012319 | -0.012549 | 1.370031 | 0.000636 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000643
|
BRD-K11640013-236-10-1
|
ACH-000207
|
DETROIT562_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 1.328641 | 0.006416 | -0.098728 | 1.168349 | 0.000037 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000207
|
BRD-K11640013-236-10-1
|
ACH-000260
|
SKNAS_AUTONOMIC_GANGLIA
|
HTS002
| 1 | 1.675899 | 0.048022 | -0.012482 | 1.407842 | 0.000012 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000260
|
BRD-K11640013-236-10-1
|
ACH-000019
|
MCF7_BREAST
|
HTS002
| 1 | 2.039194 | -0.061396 | -0.011421 | 1.449019 | 0.000881 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000019
|
BRD-K11640013-236-10-1
|
ACH-000582
|
COLO741_SKIN
|
HTS002
| 1 | 2.622021 | -0.307584 | 0.060421 | 1.520623 | 0.004513 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000582
|
BRD-K11640013-236-10-1
|
ACH-000990
|
HEC108_ENDOMETRIUM
|
HTS002
| 1 | 1.596364 | -0.106401 | -0.08521 | 1.437576 | 1,302.03451 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000990
|
BRD-K11640013-236-10-1
|
ACH-000592
|
TM31_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.522219 | -0.133265 | -0.048012 | 1.361967 | 43.169256 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000592
|
BRD-K11640013-236-10-1
|
ACH-000368
|
SNU1105_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.710412 | -0.228168 | 0.073485 | 1.26555 | 0.006526 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000368
|
BRD-K11640013-236-10-1
|
ACH-000517
|
SNU410_PANCREAS
|
HTS002
| 1 | 2.506615 | -0.238916 | 0.192027 | 1.59179 | 0.010368 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000517
|
BRD-K11640013-236-10-1
|
ACH-000374
|
HCC1143_BREAST
|
HTS002
| 1 | 1.729673 | -0.039587 | -0.009101 | 1.327506 | 0.000429 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000374
|
BRD-K11640013-236-10-1
|
ACH-000527
|
OVISE_OVARY
|
HTS002
| 1 | 2.255873 | -0.122689 | -0.089375 | 1.466053 | 0.000937 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000527
|
BRD-K11640013-236-10-1
|
ACH-000759
|
MDAMB175VII_BREAST
|
HTS002
| 1 | 1.530551 | 0.426097 | -0.006834 | 1.053835 | 43.534886 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000759
|
BRD-K11640013-236-10-1
|
ACH-000308
|
EFO21_OVARY
|
HTS002
| 1 | 1.652453 | -0.177627 | 0.000033 | 1.323686 | 0.071181 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000308
|
BRD-K11640013-236-10-1
|
ACH-000991
|
SNU81_LARGE_INTESTINE
|
HTS002
| 1 | 1.928496 | 0.150356 | 0.005524 | 1.29122 | 17.755374 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000991
|
BRD-K11640013-236-10-1
|
ACH-000948
|
2313287_STOMACH
|
HTS002
| 1 | 1.291818 | 2.100297 | 0.051299 | 1.170102 | 0.034943 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000948
|
BRD-K11640013-236-10-1
|
ACH-000481
|
NCIH2170_LUNG
|
HTS002
| 1 | 1.919622 | -0.091373 | 0.020651 | 1.415666 | 0.009171 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000481
|
BRD-K11640013-236-10-1
|
ACH-000159
|
OSRC2_KIDNEY
|
HTS002
| 1 | 1.49102 | -0.285406 | 0.06186 | 1.164295 | 0.004912 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000159
|
BRD-K11640013-236-10-1
|
ACH-000929
|
NCIH2110_LUNG
|
HTS002
| 1 | 2.028129 | -0.075974 | 0.053394 | 1.466003 | 0.006437 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000929
|
BRD-K11640013-236-10-1
|
ACH-000118
|
HUPT3_PANCREAS
|
HTS002
| 1 | 2.715654 | -0.25768 | 0.114363 | 1.584444 | 0.004402 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000118
|
BRD-K11640013-236-10-1
|
ACH-000482
|
RERFLCKJ_LUNG
|
HTS002
| 1 | 1.822825 | -0.32682 | -0.114207 | 1.399962 | 0.063666 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000482
|
BRD-K11640013-236-10-1
|
ACH-000352
|
HCC1428_BREAST
|
HTS002
| 1 | 1.504085 | -1.021279 | -0.071255 | 1.154965 | 0.011506 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000352
|
BRD-K11640013-236-10-1
|
ACH-000900
|
NCIH23_LUNG
|
HTS002
| 1 | 2.062113 | -0.062112 | 0.020996 | 1.594182 | 3.762811 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000900
|
BRD-K11640013-236-10-1
|
ACH-000479
|
KNS81_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 5.170279 | -0.242485 | 0.071854 | 1.546843 | 0.000016 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000479
|
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