broad_id
string | depmap_id
string | ccle_name
string | screen_id
string | upper_limit
int64 | lower_limit
float64 | slope
float64 | r2
float64 | auc
float64 | ec50
float64 | ic50
float64 | name
string | moa
string | target
string | disease.area
string | indication
string | smiles
string | phase
string | passed_str_profiling
bool | row_name
string |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
BRD-K11640013-236-10-1
|
ACH-000748
|
SJSA1_BONE
|
HTS002
| 1 | 1.570486 | -0.006316 | -0.002873 | 1.300272 | 1,398,664.842299 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000748
|
BRD-K11640013-236-10-1
|
ACH-000788
|
A2058_SKIN
|
HTS002
| 1 | 1.343465 | -0.007497 | -0.052362 | 1.178792 | 4,552.992924 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000788
|
BRD-K11640013-236-10-1
|
ACH-000545
|
VMCUB1_URINARY_TRACT
|
HTS002
| 1 | 4.720265 | -0.477336 | 0.496101 | 2.058156 | 0.005425 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000545
|
BRD-K11640013-236-10-1
|
ACH-000762
|
YD38_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 1.820771 | 0.033788 | -0.02956 | 1.395095 | 0.71315 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000762
|
BRD-K11640013-236-10-1
|
ACH-000792
|
BFTC909_KIDNEY
|
HTS002
| 1 | 2.348876 | 0.07436 | -0.0167 | 1.851796 | 0.000052 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000792
|
BRD-K11640013-236-10-1
|
ACH-000211
|
DAOY_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 2.081878 | -0.195488 | -0.134643 | 1.261295 | 0.000152 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000211
|
BRD-K11640013-236-10-1
|
ACH-000936
|
EFO27_OVARY
|
HTS002
| 1 | 1.768761 | -0.13358 | -0.059246 | 1.265288 | 0.000549 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000936
|
BRD-K11640013-236-10-1
|
ACH-000882
|
IGR1_SKIN
|
HTS002
| 1 | 1.416803 | -0.093688 | -0.035356 | 1.139196 | 0.000044 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000882
|
BRD-K11640013-236-10-1
|
ACH-000471
|
LI7_LIVER
|
HTS002
| 1 | 2.537399 | -0.559847 | -0.05591 | 1.33747 | 0.002763 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000471
|
BRD-K11640013-236-10-1
|
ACH-000670
|
SBC5_LUNG
|
HTS002
| 1 | 1.702771 | -0.092261 | 0.151061 | 1.355831 | 0.103247 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000670
|
BRD-K11640013-236-10-1
|
ACH-000048
|
TOV112D_OVARY
|
HTS002
| 1 | 2.235971 | 0.052166 | -0.097095 | 1.270528 | 3,421,368,140.7498 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000048
|
BRD-K11640013-236-10-1
|
ACH-000599
|
PATU8902_PANCREAS
|
HTS002
| 1 | 1.604991 | -0.16538 | 0.104501 | 1.26978 | 0.019605 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000599
|
BRD-K11640013-236-10-1
|
ACH-000716
|
TT2609C02_THYROID
|
HTS002
| 1 | 1.579399 | -0.149435 | 0.168882 | 1.265853 | 0.024687 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000716
|
BRD-K11640013-236-10-1
|
ACH-000347
|
QGP1_PANCREAS
|
HTS002
| 1 | 1.737003 | -0.136331 | 0.067893 | 1.258919 | 0.000742 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000347
|
BRD-K11640013-236-10-1
|
ACH-000566
|
SW1710_URINARY_TRACT
|
HTS002
| 1 | 1.328712 | 0.078154 | -0.045634 | 1.17415 | 0.016666 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000566
|
BRD-K11640013-236-10-1
|
ACH-001016
|
BECKER_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.453394 | -0.070394 | 0.021298 | 1.199903 | 0.002591 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-001016
|
BRD-K11640013-236-10-1
|
ACH-000395
|
NCIH520_LUNG
|
HTS002
| 1 | 1.579754 | -0.013318 | -0.000497 | 1.277735 | 0.000144 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000395
|
BRD-K11640013-236-10-1
|
ACH-000407
|
SNU685_ENDOMETRIUM
|
HTS002
| 1 | 1.868024 | 0.015748 | -0.007073 | 1.422946 | 1.995689 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000407
|
BRD-K11640013-236-10-1
|
ACH-000418
|
SW1353_BONE
|
HTS002
| 1 | 1.725629 | -0.037183 | -0.096903 | 1.509338 | 835,451,288.825851 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000418
|
BRD-K11640013-236-10-1
|
ACH-000008
|
A101D_SKIN
|
HTS002
| 1 | 1.5507 | -0.162473 | 0.019297 | 1.270307 | 0.061638 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000008
|
BRD-K11640013-236-10-1
|
ACH-000191
|
BHT101_THYROID
|
HTS002
| 1 | 1.652548 | -0.279261 | 0.063441 | 1.386762 | 0.364512 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000191
|
BRD-K11640013-236-10-1
|
ACH-000941
|
HEC1B_ENDOMETRIUM
|
HTS002
| 1 | 1.467999 | 0.454789 | -0.058283 | 1.307403 | 0.011187 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000941
|
BRD-K11640013-236-10-1
|
ACH-000532
|
SNU61_LARGE_INTESTINE
|
HTS002
| 1 | 2.568234 | 0.030086 | -0.008068 | 1.678419 | 653.419674 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000532
|
BRD-K11640013-236-10-1
|
ACH-000316
|
SNU886_LIVER
|
HTS002
| 1 | 1.974259 | -0.054134 | 0.014077 | 1.446474 | 0.00349 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000316
|
BRD-K11640013-236-10-1
|
ACH-000677
|
SW1573_LUNG
|
HTS002
| 1 | 1.303922 | 0.066128 | -0.068309 | 1.163951 | 0.007003 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000677
|
BRD-K11640013-236-10-1
|
ACH-000375
|
G402_SOFT_TISSUE
|
HTS002
| 1 | 1.574252 | -0.291841 | 0.074088 | 1.409226 | 2.804772 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000375
|
BRD-K11640013-236-10-1
|
ACH-000965
|
RL952_ENDOMETRIUM
|
HTS002
| 1 | 2.165268 | -0.172734 | -0.023048 | 1.552209 | 0.041187 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000965
|
BRD-K11640013-236-10-1
|
ACH-000210
|
CADOES1_BONE
|
HTS002
| 1 | 1.987543 | 0.064314 | -0.027784 | 1.494207 | 0.075994 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000210
|
BRD-K11640013-236-10-1
|
ACH-000803
|
COLO668_LUNG
|
HTS002
| 1 | 1.445462 | -0.911952 | -0.128392 | 1.197557 | 0.044524 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000803
|
BRD-K11640013-236-10-1
|
ACH-000007
|
LS513_LARGE_INTESTINE
|
HTS002
| 1 | 2.334933 | -0.044349 | 0.053668 | 1.629572 | 0.005961 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000007
|
BRD-K11640013-236-10-1
|
ACH-000719
|
RMGI_OVARY
|
HTS002
| 1 | 1.7251 | -0.010518 | -0.017464 | 1.398949 | 16,359,764.137068 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000719
|
BRD-K11640013-236-10-1
|
ACH-000433
|
CAKI1_KIDNEY
|
HTS002
| 1 | 2.559507 | -0.087884 | 0.028576 | 1.571884 | 0.000142 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000433
|
BRD-K11640013-236-10-1
|
ACH-000688
|
OV7_OVARY
|
HTS002
| 1 | 1.776975 | 0.278434 | -0.041855 | 1.675751 | 0.000039 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000688
|
BRD-K11640013-236-10-1
|
ACH-000351
|
MKN1_STOMACH
|
HTS002
| 1 | 2.105121 | -0.041771 | 0.002091 | 1.598557 | 4.301894 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000351
|
BRD-K11640013-236-10-1
|
ACH-000627
|
LCLC103H_LUNG
|
HTS002
| 1 | 1.906716 | -0.245107 | 0.088394 | 1.353373 | 0.010192 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000627
|
BRD-K11640013-236-10-1
|
ACH-000916
|
NCIH1573_LUNG
|
HTS002
| 1 | 1.923058 | -0.188872 | 0.000233 | 1.39397 | 0.014733 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000916
|
BRD-K11640013-236-10-1
|
ACH-000863
|
DBTRG05MG_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.514707 | -0.057262 | -0.001996 | 1.248506 | 0.023322 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000863
|
BRD-K11640013-236-10-1
|
ACH-000732
|
PECAPJ41CLONED2_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 2.128061 | -0.107591 | 0.056243 | 1.544894 | 0.040981 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000732
|
BRD-K11640013-236-10-1
|
ACH-000066
|
HCC4006_LUNG
|
HTS002
| 1 | 1.343868 | -0.026973 | -0.035327 | 1.18642 | 41.33043 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000066
|
BRD-K11640013-236-10-1
|
ACH-000015
|
NCIH1581_LUNG
|
HTS002
| 1 | 1.935488 | 0.764416 | 0.082241 | 1.207218 | 1.537428 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000015
|
BRD-K11640013-236-10-1
| null | null |
HTS002
| 1 | 1.74387 | -0.008262 | -0.090997 | 1.387186 | 1,609.122311 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| false |
ACH-000511_FAILED_STR
|
BRD-K11640013-236-10-1
|
ACH-000674
|
NUGC4_STOMACH
|
HTS002
| 1 | 1.985267 | -0.046117 | -0.212307 | 1.559395 | 29.625423 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000674
|
BRD-K11640013-236-10-1
|
ACH-000892
|
NCIH1563_LUNG
|
HTS002
| 1 | 1.102714 | 0.047034 | -0.089107 | 1.061591 | 0.000014 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000892
|
BRD-K11640013-236-10-1
|
ACH-000909
|
JHUEM2_ENDOMETRIUM
|
HTS002
| 1 | 2.205135 | 0.176857 | 0.055427 | 1.400954 | 5.027419 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000909
|
BRD-K11640013-236-10-1
|
ACH-000237
|
JHOM1_OVARY
|
HTS002
| 1 | 2.056746 | -0.144566 | 0.089584 | 1.358589 | 0.00065 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000237
|
BRD-K11640013-236-10-1
|
ACH-000811
|
SKOV3_OVARY
|
HTS002
| 1 | 1.49674 | -0.259377 | 0.047488 | 1.324696 | 1.225521 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000811
|
BRD-K11640013-236-10-1
|
ACH-000312
|
SKNBE2_AUTONOMIC_GANGLIA
|
HTS002
| 1 | 1.333773 | 0.264687 | -0.212934 | 1.244167 | 0.001111 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000312
|
BRD-K11640013-236-10-1
|
ACH-000390
|
LUDLU1_LUNG
|
HTS002
| 1 | 2.444514 | -0.397323 | -0.009767 | 1.498742 | 0.009923 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000390
|
BRD-K11640013-236-10-1
|
ACH-000901
|
HCC1359_LUNG
|
HTS002
| 1 | 1.906328 | 0.01285 | -0.06552 | 1.478923 | 0.000011 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000901
|
BRD-K11640013-236-10-1
|
ACH-000307
|
PK1_PANCREAS
|
HTS002
| 1 | 1.929972 | 0.089904 | -0.116262 | 1.442597 | 0.232111 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000307
|
BRD-K11640013-236-10-1
|
ACH-000289
|
SNU466_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 2.171639 | -0.313483 | 0.041077 | 1.31667 | 0.001914 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000289
|
BRD-K11640013-236-10-1
|
ACH-000733
|
NCIH1838_LUNG
|
HTS002
| 1 | 2.07868 | -0.059717 | -0.021723 | 1.573973 | 0.683262 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000733
|
BRD-K11640013-236-10-1
|
ACH-000268
|
SNU245_BILIARY_TRACT
|
HTS002
| 1 | 2.879299 | -0.212369 | 0.002903 | 1.633507 | 0.002478 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000268
|
BRD-K11640013-236-10-1
|
ACH-000758
|
MKN74_STOMACH
|
HTS002
| 1 | 3.225806 | -0.205941 | 0.031852 | 1.343968 | 0.000012 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000758
|
BRD-K11640013-236-10-1
|
ACH-000693
|
KYSE180_OESOPHAGUS
|
HTS002
| 1 | 1.602162 | -0.079806 | 0.012034 | 1.250865 | 0.001091 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000693
|
BRD-K11640013-236-10-1
|
ACH-000684
|
KMRC1_KIDNEY
|
HTS002
| 1 | 1.798572 | -0.096188 | 0.003157 | 1.346777 | 0.004752 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000684
|
BRD-K11640013-236-10-1
|
ACH-000264
|
CALU6_LUNG
|
HTS002
| 1 | 1.852854 | -0.437989 | 0.21118 | 1.284252 | 0.009438 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000264
|
BRD-K11640013-236-10-1
|
ACH-000027
|
GOS3_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.500742 | 0.155202 | -0.048975 | 1.244565 | 0.106821 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000027
|
BRD-K11640013-236-10-1
|
ACH-000671
|
HUH6_LIVER
|
HTS002
| 1 | 1.66703 | 0.075669 | -0.081804 | 1.386377 | 0.00109 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000671
|
BRD-K11640013-236-10-1
|
ACH-000205
|
PK59_PANCREAS
|
HTS002
| 1 | 2.403623 | -0.012022 | -0.0029 | 1.717757 | 3.427865 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000205
|
BRD-K11640013-236-10-1
|
ACH-000720
|
TCCSUP_URINARY_TRACT
|
HTS002
| 1 | 2.289243 | -0.085749 | -0.079905 | 1.618924 | 0.030406 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000720
|
BRD-K11640013-236-10-1
|
ACH-000885
|
TOV21G_OVARY
|
HTS002
| 1 | 1.545941 | -0.20519 | 0.015543 | 1.158042 | 0.000705 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000885
|
BRD-K11640013-236-10-1
|
ACH-000663
|
OVTOKO_OVARY
|
HTS002
| 1 | 1.746346 | 0.173178 | 0.059748 | 1.334067 | 0.282414 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000663
|
BRD-K11640013-236-10-1
|
ACH-000647
|
TE1_OESOPHAGUS
|
HTS002
| 1 | 1.696869 | -4.645325 | 0.240101 | 1.243009 | 0.017997 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000647
|
BRD-K11640013-236-10-1
|
ACH-000243
|
DANG_PANCREAS
|
HTS002
| 1 | 1.909147 | -0.251841 | 0.085235 | 1.370121 | 0.014681 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000243
|
BRD-K11640013-236-10-1
|
ACH-000255
|
LMSU_STOMACH
|
HTS002
| 1 | 1.776721 | 0.018786 | -0.012221 | 1.40648 | 0.00054 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000255
|
BRD-K11640013-236-10-1
|
ACH-000335
|
MSTO211H_PLEURA
|
HTS002
| 1 | 1.526085 | -3.063449 | 0.248325 | 1.278538 | 0.103972 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000335
|
BRD-K11640013-236-10-1
|
ACH-000147
|
T47D_BREAST
|
HTS002
| 1 | 1.801727 | 0.102882 | -0.011991 | 1.285448 | 27.830958 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000147
|
BRD-K11640013-236-10-1
|
ACH-000090
|
PC3_PROSTATE
|
HTS002
| 1 | 1.381487 | -0.021743 | -0.004213 | 1.192944 | 0.225963 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000090
|
BRD-K11640013-236-10-1
|
ACH-000171
|
VMRCRCZ_KIDNEY
|
HTS002
| 1 | 1.32468 | 0.064774 | -0.193365 | 1.195546 | 0.000122 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000171
|
BRD-K11640013-236-10-1
|
ACH-000614
|
RVH421_SKIN
|
HTS002
| 1 | 2.053021 | 0.078336 | -0.015774 | 1.472114 | 1.138147 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000614
|
BRD-K11640013-236-10-1
|
ACH-000132
|
JHOS2_OVARY
|
HTS002
| 1 | 2.573058 | -0.248526 | 0.103792 | 1.325946 | 0.000203 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000132
|
BRD-K11640013-236-10-1
|
ACH-000274
|
HS852T_SKIN
|
HTS002
| 1 | 1.928848 | 0.016991 | -0.040045 | 1.483502 | 0.000617 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000274
|
BRD-K11640013-236-10-1
| null | null |
HTS002
| 1 | 1.340058 | -0.121317 | -0.043999 | 1.248983 | 387.554578 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| false |
ACH-000807_FAILED_STR
|
BRD-K11640013-236-10-1
|
ACH-000343
|
NCIH522_LUNG
|
HTS002
| 1 | 2.010027 | -0.107778 | -0.000734 | 1.464893 | 0.017245 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000343
|
BRD-K11640013-236-10-1
|
ACH-000022
|
PATU8988S_PANCREAS
|
HTS002
| 1 | 2.108775 | -0.040167 | -0.108336 | 1.524799 | 0.005419 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000022
|
BRD-K11640013-236-10-1
|
ACH-000192
|
MFE280_ENDOMETRIUM
|
HTS002
| 1 | 2.689283 | -0.114968 | 0.073445 | 1.64125 | 0.000978 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000192
|
BRD-K11640013-236-10-1
|
ACH-000959
|
SNUC4_LARGE_INTESTINE
|
HTS002
| 1 | 1.988791 | -0.412552 | -0.034869 | 1.266899 | 0.003507 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000959
|
BRD-K11640013-236-10-1
| null | null |
HTS002
| 1 | 1.671785 | 0.160577 | -0.025544 | 1.239977 | 3.621317 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| false |
ACH-000028_FAILED_STR
|
BRD-K11640013-236-10-1
|
ACH-000637
|
KYSE520_OESOPHAGUS
|
HTS002
| 1 | 1.886956 | -0.062032 | 0.052697 | 1.394087 | 0.002066 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000637
|
BRD-K11640013-236-10-1
|
ACH-000968
|
COLO792_SKIN
|
HTS002
| 1 | 1.165032 | -0.026125 | -0.217952 | 1.114703 | 4,016,995,961,359.87 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000968
|
BRD-K11640013-236-10-1
|
ACH-000155
|
SW1990_PANCREAS
|
HTS002
| 1 | 1.592521 | -0.087002 | -0.045548 | 1.364647 | 18.780871 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000155
|
BRD-K11640013-236-10-1
|
ACH-000605
|
TE6_OESOPHAGUS
|
HTS002
| 1 | 2.065128 | 0.170708 | -0.003201 | 1.320984 | 13.996873 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000605
|
BRD-K11640013-236-10-1
|
ACH-000775
|
NCIH727_LUNG
|
HTS002
| 1 | 2.056065 | -0.109239 | 0.046763 | 1.49266 | 0.022229 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000775
|
BRD-K11640013-236-10-1
|
ACH-000042
|
PANC0203_PANCREAS
|
HTS002
| 1 | 1.703582 | -0.248443 | 0.073162 | 1.198526 | 0.001205 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000042
|
BRD-K11640013-236-10-1
|
ACH-000860
|
NCIH358_LUNG
|
HTS002
| 1 | 2.259654 | -0.290703 | 0.168715 | 1.55819 | 0.0314 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000860
|
BRD-K11640013-236-10-1
|
ACH-000994
|
HEC59_ENDOMETRIUM
|
HTS002
| 1 | 1.408274 | 0.063933 | -0.006196 | 1.236089 | 0.000539 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000994
|
BRD-K11640013-236-10-1
|
ACH-000277
|
HCC1419_BREAST
|
HTS002
| 1 | 2.195537 | -0.180706 | 0.057601 | 1.603237 | 0.087005 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000277
|
BRD-K11640013-236-10-1
|
ACH-000496
|
NCIH1792_LUNG
|
HTS002
| 1 | 3.02135 | 0.033188 | -0.077564 | 1.740812 | 1,173,647.150309 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000496
|
BRD-K11640013-236-10-1
|
ACH-000866
|
NCIH1048_LUNG
|
HTS002
| 1 | 2.759122 | -0.925993 | 0.181668 | 1.179237 | 0.000945 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000866
|
BRD-K11640013-236-10-1
|
ACH-000869
|
NCIH1568_LUNG
|
HTS002
| 1 | 1.370182 | -0.117593 | -0.008986 | 1.2948 | 11,148.691766 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000869
|
BRD-K11640013-236-10-1
|
ACH-000678
|
MKN7_STOMACH
|
HTS002
| 1 | 1.265321 | -0.12339 | 0.000001 | 1.215591 | 15,335.590024 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000678
|
BRD-K11640013-236-10-1
|
ACH-000493
|
SNU423_LIVER
|
HTS002
| 1 | 1.957194 | -0.199612 | 0.048525 | 1.318402 | 0.001845 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000493
|
BRD-K11640013-236-10-1
|
ACH-000468
|
PK45H_PANCREAS
|
HTS002
| 1 | 1.315691 | -0.540575 | -0.108984 | 1.188248 | 0.23209 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000468
|
BRD-K11640013-236-10-1
|
ACH-000097
|
ZR751_BREAST
|
HTS002
| 1 | 1.606101 | -0.230654 | 0.025157 | 1.237257 | 0.009516 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000097
|
BRD-K11640013-236-10-1
|
ACH-000313
|
KMRC3_KIDNEY
|
HTS002
| 1 | 1.451298 | 0.531066 | -0.051734 | 1.187159 | 0.205976 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000313
|
BRD-K11640013-236-10-1
|
ACH-000169
|
RD_SOFT_TISSUE
|
HTS002
| 1 | 2.073802 | 8.729462 | 0.594239 | 1.843694 | 0.004883 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000169
|
BRD-K11640013-236-10-1
| null | null |
HTS002
| 1 | 1.632963 | -1.688638 | 0.263893 | 1.326709 | 0.091394 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| false |
ACH-000010_FAILED_STR
|
BRD-K11640013-236-10-1
|
ACH-000895
|
CL34_LARGE_INTESTINE
|
HTS002
| 1 | 2.404562 | -1.433733 | 0.091308 | 1.711853 | 0.083476 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000895
|
BRD-K11640013-236-10-1
|
ACH-000841
|
NCIH2087_LUNG
|
HTS002
| 1 | 2.799336 | -0.184072 | -0.112432 | 1.508342 | 0.000363 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000841
|
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