broad_id
string | depmap_id
string | ccle_name
string | screen_id
string | upper_limit
int64 | lower_limit
float64 | slope
float64 | r2
float64 | auc
float64 | ec50
float64 | ic50
float64 | name
string | moa
string | target
string | disease.area
string | indication
string | smiles
string | phase
string | passed_str_profiling
bool | row_name
string |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
BRD-K11640013-236-10-1
|
ACH-000911
|
NUGC3_STOMACH
|
HTS002
| 1 | 1.742325 | 0.008433 | -0.00717 | 1.336988 | 253,882,082.147056 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000911
|
BRD-K11640013-236-10-1
|
ACH-000401
|
COLO800_SKIN
|
HTS002
| 1 | 1.428826 | 0.153416 | -0.071985 | 1.172777 | 1.139235 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000401
|
BRD-K11640013-236-10-1
|
ACH-000276
|
HCC38_BREAST
|
HTS002
| 1 | 2.188671 | -0.047405 | 0.022493 | 1.514134 | 0.000248 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000276
|
BRD-K11640013-236-10-1
|
ACH-000724
|
HT1376_URINARY_TRACT
|
HTS002
| 1 | 2.428802 | -0.139121 | -0.060668 | 1.618561 | 0.010437 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000724
|
BRD-K11640013-236-10-1
|
ACH-000092
|
NCIH2452_PLEURA
|
HTS002
| 1 | 1.263944 | -3.135204 | 0.001996 | 1.141446 | 0.110675 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000092
|
BRD-K11640013-236-10-1
|
ACH-000890
|
SW1271_LUNG
|
HTS002
| 1 | 1.826172 | -0.114797 | 0.080457 | 1.403194 | 0.050922 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000890
|
BRD-K11640013-236-10-1
| null | null |
HTS002
| 1 | 2.462477 | 0.318686 | -0.065373 | 1.495422 | 0.93797 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| false |
ACH-000539_FAILED_STR
|
BRD-K11640013-236-10-1
|
ACH-000800
|
NCIH446_LUNG
|
HTS002
| 1 | 3.301652 | -0.399445 | 0.219805 | 1.33952 | 0.00035 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000800
|
BRD-K11640013-236-10-1
|
ACH-000899
|
WM88_SKIN
|
HTS002
| 1 | 1.717667 | -0.113718 | 0.059756 | 1.267428 | 0.000715 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000899
|
BRD-K11640013-236-10-1
|
ACH-000996
|
HEC251_ENDOMETRIUM
|
HTS002
| 1 | 1.763204 | -0.05625 | -0.00604 | 1.732489 | 294,344,917,941,530,000,000,000 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000996
|
BRD-K11640013-236-10-1
|
ACH-000622
|
KNS42_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.742762 | -0.088329 | -0.077459 | 1.502982 | 387.634374 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000622
|
BRD-K11640013-236-10-1
|
ACH-000403
|
NCIH747_LARGE_INTESTINE
|
HTS002
| 1 | 13.478075 | -2.883474 | -0.292917 | 1.025313 | 0.000228 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000403
|
BRD-K11640013-236-10-1
|
ACH-000988
|
MFE319_ENDOMETRIUM
|
HTS002
| 1 | 1.387233 | 0.279765 | -0.101377 | 1.301818 | 0.000475 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000988
|
BRD-K11640013-236-10-1
|
ACH-000848
|
JHH7_LIVER
|
HTS002
| 1 | 2.542588 | -0.075311 | 0.063643 | 1.6724 | 0.002451 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000848
|
BRD-K11640013-236-10-1
|
ACH-000785
|
NCIH2126_LUNG
|
HTS002
| 1 | 2.144866 | 0.009103 | -0.041305 | 1.582871 | 0.00142 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000785
|
BRD-K11640013-236-10-1
|
ACH-000544
|
OE21_OESOPHAGUS
|
HTS002
| 1 | 2.338012 | -0.116706 | 0.154566 | 1.606745 | 0.015126 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000544
|
BRD-K11640013-236-10-1
|
ACH-000982
|
GP2D_LARGE_INTESTINE
|
HTS002
| 1 | 1.517236 | 0.138608 | -0.018511 | 1.347355 | 0.000373 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000982
|
BRD-K11640013-236-10-1
|
ACH-000021
|
NCIH1693_LUNG
|
HTS002
| 1 | 2.57977 | -0.133631 | -0.001285 | 1.388586 | 0.000014 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000021
|
BRD-K11640013-236-10-1
|
ACH-000823
|
KYSE140_OESOPHAGUS
|
HTS002
| 1 | 1.854672 | 0.154524 | -0.120699 | 1.361603 | 0.637468 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000823
|
BRD-K11640013-236-10-1
|
ACH-000915
|
IPC298_SKIN
|
HTS002
| 1 | 2.063993 | -0.02029 | -0.004045 | 1.513931 | 0.002738 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000915
|
BRD-K11640013-236-10-1
|
ACH-000984
|
HEC6_ENDOMETRIUM
|
HTS002
| 1 | 1.790365 | -0.022289 | 0.00339 | 1.390236 | 0.025384 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000984
|
BRD-K11640013-236-10-1
|
ACH-001306
|
8305C_THYROID
|
HTS002
| 1 | 1.805802 | 3.123882 | -0.088153 | 1.212696 | 0.772014 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-001306
|
BRD-K11640013-236-10-1
|
ACH-000318
|
TE10_OESOPHAGUS
|
HTS002
| 1 | 1.923952 | -0.041594 | 0.028404 | 1.502877 | 5.659461 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000318
|
BRD-K11640013-236-10-1
|
ACH-000840
|
HCC366_LUNG
|
HTS002
| 1 | 2.216253 | -0.229021 | 0.084227 | 1.382107 | 0.001864 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000840
|
BRD-K11640013-236-10-1
|
ACH-000503
|
BICR16_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 1.233264 | -0.006434 | -0.151949 | 1.121323 | 21,174.724243 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000503
|
BRD-K11640013-236-10-1
|
ACH-000919
|
IM95_STOMACH
|
HTS002
| 1 | 1.218268 | 0.133396 | -0.08628 | 1.125062 | 0.007992 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000919
|
BRD-K11640013-236-10-1
|
ACH-000188
|
SCC25_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 3.445623 | -5.209864 | 0.400937 | 1.124365 | 0.000985 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000188
|
BRD-K11640013-236-10-1
|
ACH-000618
|
SNU1041_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 1.403244 | -0.28039 | 0.003324 | 1.243888 | 0.445687 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000618
|
BRD-K11640013-236-10-1
|
ACH-000822
|
SKMEL24_SKIN
|
HTS002
| 1 | 1.921665 | -0.135421 | -0.017939 | 1.607571 | 12.066916 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000822
|
BRD-K11640013-236-10-1
|
ACH-000292
|
NCIH841_LUNG
|
HTS002
| 1 | 1.608445 | -0.004894 | 0.002093 | 1.306102 | 0.975766 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000292
|
BRD-K11640013-236-10-1
|
ACH-000827
|
WM793_SKIN
|
HTS002
| 1 | 1.972202 | -0.137893 | 0.13984 | 1.42572 | 0.011949 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000827
|
BRD-K11640013-236-10-1
|
ACH-000411
|
769P_KIDNEY
|
HTS002
| 1 | 1.653722 | -0.211744 | 0.039638 | 1.354371 | 0.18565 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000411
|
BRD-K11640013-236-10-1
|
ACH-000139
|
PANC0327_PANCREAS
|
HTS002
| 1 | 1.478238 | -0.349491 | -0.162901 | 1.124212 | 0.002091 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000139
|
BRD-K11640013-236-10-1
|
ACH-000569
|
ISTMES1_PLEURA
|
HTS002
| 1 | 1.6241 | -0.304996 | 0.117535 | 1.174331 | 0.002105 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000569
|
BRD-K11640013-236-10-1
|
ACH-000741
|
UBLC1_URINARY_TRACT
|
HTS002
| 1 | 2.221246 | -0.154455 | 0.028543 | 1.524236 | 0.011349 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000741
|
BRD-K11640013-236-10-1
|
ACH-000425
|
UACC62_SKIN
|
HTS002
| 1 | 1.678938 | -0.144227 | 0.008588 | 1.383832 | 0.520225 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000425
|
BRD-K11640013-236-10-1
|
ACH-000231
|
KALS1_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.669699 | 0.13857 | -0.003198 | 1.244491 | 4.902338 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000231
|
BRD-K11640013-236-10-1
|
ACH-000730
|
SKMEL5_SKIN
|
HTS002
| 1 | 2.512472 | -0.209369 | 0.052569 | 1.715111 | 0.044451 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000730
|
BRD-K11640013-236-10-1
|
ACH-000500
|
SNU46_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 1.709904 | 0.009507 | -0.004399 | 1.354311 | 0.11427 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000500
|
BRD-K11640013-236-10-1
|
ACH-000222
|
ASPC1_PANCREAS
|
HTS002
| 1 | 1.271259 | -0.348013 | 0.01484 | 1.109583 | 0.019897 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000222
|
BRD-K11640013-236-10-1
|
ACH-000477
|
MALME3M_SKIN
|
HTS002
| 1 | 2.514879 | -0.240516 | -0.081082 | 1.39866 | 0.000699 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000477
|
BRD-K11640013-236-10-1
|
ACH-000223
|
HCC1937_BREAST
|
HTS002
| 1 | 2.273166 | -0.105433 | 0.120765 | 1.520524 | 0.002194 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000223
|
BRD-K11640013-236-10-1
|
ACH-000495
|
TUHR4TKB_KIDNEY
|
HTS002
| 1 | 1.612385 | 0.00605 | -0.00314 | 1.292157 | 301,158.271176 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000495
|
BRD-K11640013-236-10-1
|
ACH-000434
|
NCIH1915_LUNG
|
HTS002
| 1 | 2.067909 | -0.140243 | 0.222552 | 1.517429 | 0.049398 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000434
|
BRD-K11640013-236-10-1
|
ACH-000744
|
NCIH1623_LUNG
|
HTS002
| 1 | 1.814873 | -0.048374 | -0.042133 | 1.44451 | 3.456481 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000744
|
BRD-K11640013-236-10-1
|
ACH-000107
|
CAPAN2_PANCREAS
|
HTS002
| 1 | 1.783144 | -0.016597 | -0.081395 | 1.386879 | 0.018416 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000107
|
BRD-K11640013-236-10-1
|
ACH-000516
|
CAL78_BONE
|
HTS002
| 1 | 1.482942 | -0.099956 | -0.008055 | 1.310416 | 31.132771 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000516
|
BRD-K11640013-236-10-1
|
ACH-000898
|
SNU719_STOMACH
|
HTS002
| 1 | 1.901386 | -0.948598 | -0.170149 | 1.07749 | 0.000744 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000898
|
BRD-K11640013-236-10-1
|
ACH-000040
|
U118MG_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.395775 | 0.057622 | -0.124835 | 1.230437 | 0.000237 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000040
|
BRD-K11640013-236-10-1
|
ACH-000808
|
HUH28_BILIARY_TRACT
|
HTS002
| 1 | 1.735065 | 0.144829 | -0.008232 | 1.513037 | 0.000193 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000808
|
BRD-K11640013-236-10-1
|
ACH-000447
|
NCIH2228_LUNG
|
HTS002
| 1 | 1.888692 | -0.289845 | -0.049418 | 1.300278 | 0.005373 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000447
|
BRD-K11640013-236-10-1
|
ACH-000715
|
SNU1214_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 2.426601 | -0.333958 | 0.051915 | 1.371671 | 0.001892 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000715
|
BRD-K11640013-236-10-1
|
ACH-000542
|
HEYA8_OVARY
|
HTS002
| 1 | 1.813496 | 0.177279 | -0.06342 | 1.542573 | 0.001236 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000542
|
BRD-K11640013-236-10-1
|
ACH-000943
|
RKO_LARGE_INTESTINE
|
HTS002
| 1 | 2.184781 | -2.014774 | 0.566324 | 1.478107 | 0.030633 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000943
|
BRD-K11640013-236-10-1
|
ACH-000174
|
CAL62_THYROID
|
HTS002
| 1 | 1.08041 | 0.207004 | -0.125661 | 1.043671 | 0.031639 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000174
|
BRD-K11640013-236-10-1
|
ACH-000018
|
T24_URINARY_TRACT
|
HTS002
| 1 | 1.381381 | -0.032212 | -0.011326 | 1.205718 | 10.629571 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000018
|
BRD-K11640013-236-10-1
|
ACH-000906
|
ES2_OVARY
|
HTS002
| 1 | 1.195965 | 0.131904 | -0.045776 | 1.110495 | 0.010441 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000906
|
BRD-K11640013-236-10-1
|
ACH-000784
|
KYSE70_OESOPHAGUS
|
HTS002
| 1 | 2.424162 | -0.062399 | 0.035549 | 1.703436 | 0.052783 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000784
|
BRD-K11640013-236-10-1
|
ACH-000265
|
KP4_PANCREAS
|
HTS002
| 1 | 2.303569 | 0.049874 | -0.012282 | 1.547013 | 53.755604 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000265
|
BRD-K11640013-236-10-1
|
ACH-000880
|
AGS_STOMACH
|
HTS002
| 1 | 1.700504 | 0.173693 | -0.33678 | 1.390491 | 0.019148 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000880
|
BRD-K11640013-236-10-1
|
ACH-000961
|
ISHIKAWAHERAKLIO02ER_ENDOMETRIUM
|
HTS002
| 1 | 1.821714 | 5.306218 | 0.665271 | 1.242334 | 0.571622 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000961
|
BRD-K11640013-236-10-1
|
ACH-000847
|
HGC27_STOMACH
|
HTS002
| 1 | 3.296311 | -0.001513 | -0.021917 | 2.148976 | 0.200934 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000847
|
BRD-K11640013-236-10-1
|
ACH-000896
|
647V_URINARY_TRACT
|
HTS002
| 1 | 1.804133 | -0.329293 | 0.283189 | 1.480576 | 0.330803 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000896
|
BRD-K11640013-236-10-1
|
ACH-000685
|
L33_PANCREAS
|
HTS002
| 1 | 2.701044 | -0.203817 | 0.00117 | 1.359329 | 0.000077 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000685
|
BRD-K11640013-236-10-1
|
ACH-000376
|
SF295_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.741625 | 0.04539 | -0.039632 | 1.379844 | 0.02659 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000376
|
BRD-K11640013-236-10-1
|
ACH-000428
|
UO31_KIDNEY
|
HTS002
| 1 | 1.615317 | 0.103748 | -0.038586 | 1.36886 | 0.001479 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000428
|
BRD-K11640013-236-10-1
|
ACH-000749
|
DMS273_LUNG
|
HTS002
| 1 | 1.662471 | -0.941338 | 0.098157 | 1.313593 | 0.060002 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000749
|
BRD-K11640013-236-10-1
|
ACH-000572
|
G361_SKIN
|
HTS002
| 1 | 2.156269 | -0.333037 | 0.00194 | 1.583778 | 0.083861 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000572
|
BRD-K11640013-236-10-1
|
ACH-000704
|
OAW42_OVARY
|
HTS002
| 1 | 1.683148 | 0.053795 | 0.003766 | 1.322146 | 0.656685 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000704
|
BRD-K11640013-236-10-1
|
ACH-000457
|
CAL54_KIDNEY
|
HTS002
| 1 | 1.023381 | 0.077887 | -0.131089 | 1.012647 | 0.009283 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000457
|
BRD-K11640013-236-10-1
|
ACH-000601
|
MIAPACA2_PANCREAS
|
HTS002
| 1 | 1.870897 | -0.099036 | 0.084304 | 1.393215 | 0.010548 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000601
|
BRD-K11640013-236-10-1
|
ACH-000651
|
SW620_LARGE_INTESTINE
|
HTS002
| 1 | 1.923264 | -0.135548 | 0.13516 | 1.377179 | 0.004626 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000651
|
BRD-K11640013-236-10-1
|
ACH-000361
|
SKHEP1_LIVER
|
HTS002
| 1 | 1.628982 | -1.200554 | 0.220914 | 1.321809 | 0.087521 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000361
|
BRD-K11640013-236-10-1
|
ACH-000570
|
YKG1_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 3.121977 | -1.425146 | 0.045865 | 1.142181 | 0.000821 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000570
|
BRD-K11640013-236-10-1
|
ACH-000396
|
J82_URINARY_TRACT
|
HTS002
| 1 | 1.576697 | 0.041711 | -0.01769 | 1.328322 | 0.000095 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000396
|
BRD-K11640013-236-10-1
|
ACH-000777
|
KYSE30_OESOPHAGUS
|
HTS002
| 1 | 1.808593 | -0.317588 | 0.089095 | 1.247199 | 0.003713 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000777
|
BRD-K11640013-236-10-1
|
ACH-000096
|
G401_SOFT_TISSUE
|
HTS002
| 1 | 1.353683 | -0.088723 | -0.067786 | 1.304453 | 83,190,199.302443 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000096
|
BRD-K11640013-236-10-1
|
ACH-000940
|
AN3CA_ENDOMETRIUM
|
HTS002
| 1 | 0.759295 | 7.660707 | -0.017661 | 0.879321 | 0.077103 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000940
|
BRD-K11640013-236-10-1
|
ACH-001318
|
PLCPRF5_LIVER
|
HTS002
| 1 | 2.420398 | -0.339289 | 0.00014 | 1.362089 | 0.001782 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-001318
|
BRD-K11640013-236-10-1
|
ACH-000332
|
YAPC_PANCREAS
|
HTS002
| 1 | 1.684774 | -0.025911 | 0.0102 | 1.338774 | 0.034555 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000332
|
BRD-K11640013-236-10-1
|
ACH-000839
|
SCABER_URINARY_TRACT
|
HTS002
| 1 | 1.490566 | -1.561814 | 0.259584 | 1.426867 | 3.123285 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000839
|
BRD-K11640013-236-10-1
|
ACH-000082
|
G292CLONEA141B1_BONE
|
HTS002
| 1 | 1.38241 | 0.248167 | -0.049755 | 1.243593 | 0.006247 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000082
|
BRD-K11640013-236-10-1
|
ACH-000421
|
SW837_LARGE_INTESTINE
|
HTS002
| 1 | 2.749835 | 0.199612 | 0.076928 | 1.441168 | 26.543523 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000421
|
BRD-K11640013-236-10-1
|
ACH-000524
|
KURAMOCHI_OVARY
|
HTS002
| 1 | 1.385307 | -0.018517 | -0.037472 | 1.218361 | 156,303.700508 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000524
|
BRD-K11640013-236-10-1
|
ACH-000469
|
YH13_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.50019 | 0.005796 | -0.097309 | 1.199275 | 597,054,837,825,749,000,000,000,000,000 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000469
|
BRD-K11640013-236-10-1
|
ACH-000153
|
NCIH2052_PLEURA
|
HTS002
| 1 | 3.597283 | -1.049127 | 0.00651 | 1.274905 | 0.001147 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000153
|
BRD-K11640013-236-10-1
|
ACH-000805
|
COLO679_SKIN
|
HTS002
| 1 | 1.243172 | -0.046431 | -0.046801 | 1.137939 | 27.217531 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000805
|
BRD-K11640013-236-10-1
|
ACH-000429
|
A704_KIDNEY
|
HTS002
| 1 | 2.840002 | -1.038049 | 0.207524 | 1.182817 | 0.00103 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000429
|
BRD-K11640013-236-10-1
|
ACH-000108
|
KP3_PANCREAS
|
HTS002
| 1 | 1.693096 | 0.060108 | -0.04867 | 1.364568 | 0.013658 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000108
|
BRD-K11640013-236-10-1
|
ACH-000939
|
SKUT1_SOFT_TISSUE
|
HTS002
| 1 | 1.766718 | -0.051606 | -0.036032 | 1.364738 | 0.011758 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000939
|
BRD-K11640013-236-10-1
|
ACH-000323
|
42MGBA_CENTRAL_NERVOUS_SYSTEM
|
HTS002
| 1 | 1.522701 | -1.599255 | 0.305426 | 1.26317 | 0.08081 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000323
|
BRD-K11640013-236-10-1
|
ACH-000219
|
A375_SKIN
|
HTS002
| 1 | 1.549595 | -0.067671 | -0.188216 | 1.261863 | 0.019176 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000219
|
BRD-K11640013-236-10-1
|
ACH-000903
|
FTC133_THYROID
|
HTS002
| 1 | 1.571152 | -0.06117 | -0.00306 | 1.274131 | 0.020855 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000903
|
BRD-K11640013-236-10-1
|
ACH-000054
|
HT1080_SOFT_TISSUE
|
HTS002
| 1 | 2.099609 | -0.05529 | 0.007646 | 1.642697 | 38.782425 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000054
|
BRD-K11640013-236-10-1
|
ACH-000302
|
SNU1077_ENDOMETRIUM
|
HTS002
| 1 | 2.318705 | -0.119936 | -0.014304 | 1.599594 | 0.016451 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000302
|
BRD-K11640013-236-10-1
|
ACH-000324
|
JHOC5_OVARY
|
HTS002
| 1 | 1.283096 | -0.003692 | -0.071351 | 1.14063 | 0.002328 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000324
|
BRD-K11640013-236-10-1
|
ACH-000164
|
PANC1_PANCREAS
|
HTS002
| 1 | 2.998659 | -0.216914 | -0.076756 | 1.426407 | 0.000118 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000164
|
BRD-K11640013-236-10-1
|
ACH-000549
|
SNU1076_UPPER_AERODIGESTIVE_TRACT
|
HTS002
| 1 | 1.798924 | -0.568977 | -0.021623 | 1.26019 | 0.010929 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000549
|
BRD-K11640013-236-10-1
|
ACH-000650
|
IGR37_SKIN
|
HTS002
| 1 | 1.340513 | -0.23931 | 0.097515 | 1.207073 | 0.597607 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000650
|
BRD-K11640013-236-10-1
|
ACH-000217
|
JHH6_LIVER
|
HTS002
| 1 | 2.357832 | 0.011958 | -0.006512 | 1.68449 | 0.019784 | null |
sulfamethazine
|
PABA antagonist
| null |
gastroenterology
|
enteritis, enteritis
|
Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1, Cc1cc(C)nc(NS(=O)(=O)c2ccc(N)cc2)n1
|
Launched
| true |
ACH-000217
|
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